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T ? ????????藿h? ?T ???TTr??ff?乔??????? ___PPT10????iOv+q?D?' y????= @B D?' ?????= @BA?%?( < +O%?( < +D?' =%(????D?' =%(D袼' =?@B?B?BB0B%(D聒' =1?:Bvisible*?3>?B?style.visibility<?T????????%(D' =+褓4 8??CB#ppt_xBCB#ppt_xB*?3>B ppt_x<?T????????D' =+襻4 8??CB1+#ppt_h/2BCB#ppt_yB*?3>B ppt_y<?T????????+8+0+T0 +T?0 {?囗X ?  X X  ???????? ??????"??.t ??Section 2 Chloramphenicol&?$`  X  ???????? ??????"????  ???00 Antibacterial action0 &? f3? X ?????? ??????"??P??? ??x?0___PPT10??8___PPT9? ??Chloramphenicol is either bacteriostatic or bactericidal It is active against both aerobic and anaerobic gram-positive and gram-negative organisms It has effective against rickettsiae, helicoids, Chlamydia and mycoplasma.  ?&?ffH ?   @`??? X ? ????????藿h? ? ???33?洙??33???y___PPT10?Y+D?' ????= @B +??0 ?疰AKK\?A?  \??  y@  \ ? ? \? ? G???0e???0e??????    B8CDE?F??????? ?? 5%狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??A?BCD|E???????H00P?0`XP??Hx??xP(80(?P0@        ?S"?????? X{ ? \ ? ?;?0e???0e??????    BC`DE?F???ff??? ff? 5%狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??A?BCD|E?????%%?8`$D(?pH 8X? P`?p?xpPh?H@ 8?8@H0`?p????8 0@            ?S"???????? @ 瘌2 \? 3 ??@??????f??8c?????#" `??6]  ?? 疠 \ ???????览 ?????"??J? f  ??P '?f3黏2 \  ?????3烫8c?????#" `??K)e 疸 \ ??dh???览 ?????#" `??j? f  ??A '?f3?  \ ?????f?????"?? c y ?  \ ???????????"??*c ? ?  \ ???????????"???c  ?  \ ???????????"??c / ?  \ ???????????"??/c ? ? \ ???????????"???c  ? \ ???????????"??c 7 甬? @+& \C# ?9^! ? \ ?泯????f?????"???&? \  ?泯??????????"??#? \  ?泯??????????"??T?? \  ?泯??????????"???\痂?  ? ' \# ?3穰 \ 3 ?泯B C<DE连F??????? ??++??vP.1)?6?Glkp?g?d^^??6 *I'PQ^gs??????<"+H<Q6[2c*j"lt??  @              ?"` ? '鹬 \ 3 ?泯BCPDEF?????? ??? /P@ ?"` ? 鹑2 \ c ?泯??????????????? @?????#"  `??@+甬? @+& \C# ? R ? \ ?泯????f?????"???&? \  ?泯??????????"??#? \  ?泯??????????"??T?? \  ?泯??????????"???\痂?  ? ' \# ?3穰 \ 3 ?泯B C<DE连F??????? ??++??vP.1)?6?Glkp?g?d^^??6 *I'PQ^gs??????<"+H<Q6[2c*j"lt??  @              ?"` ? '鹬  \ 3 ?泯BCPDEF?????? ??? /P@ ?"` ? 鹑2 !\ c ?泯??????????????? @?????#"  `??@+??  @ "\ ?0x ?$D 0? #\? ? G???0e???0e??????    B8CDE?F??????? ?? 5%狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??A?BCD|E???????H00P?0`XP??Hx??xP(80(?P0@        ?S"??????  ? $\ ? ?;?0e???0e??????    BC`DE?F???ff??? ff? 5%狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??A?BCD|E?????%%?8`$D(?pH 8X? P`?p?xpPh?H@ 8?8@H0`?p????8 0@            ?S"??????^ z瘌2 %\? 3 ?????????f??8c?????#" `??9  ?? 疠 &\ ??????览 ?????"??  ??P '?f3黏2 '\  ?????3烫8c?????#" `??A 疸 (\ ??啾???览 ?????#" `??5  ??A '?f3? )\ ?????f?????"?? @6? *\ ???????????"?? K6? +\ ???????????"??K 6? ,\ ???????????"??? 6? -\ ???????????"?? Q6? .\ ???????????"??O 6? /\ ???????????"?? 6疖? ? @?  0\?# ? ,? 皎? @+& 1\ ?? @@ ? 2\ ?泯????f?????"???&? 3\  ?泯??????????"??#? 4\  ?泯??????????"??T?? 5\  ?泯??????????"???\痂?  ? ' 6\# ?3穰 7\ 3 ?泯B C<DE连F??????? ??++??vP.1)?6?Glkp?g?d^^??6 *I'PQ^gs??????<"+H<Q6[2c*j"lt??  @              ?"` ? '鹬 8\ 3 ?泯BCPDEF?????? ??? /P@ ?"` ? 鹑2 9\ c ?泯??????????????? @?????#"  `??@+鹑2 :\B c ?泯??????????????? @?????#"  `?? `? 鹭? @ h X #  ;\ ? ? ? <\B ?泯????f?????"??@ X ! ? =\B  ?泯??????????"??C ? ? >\B  ?泯??????????"??? ! ? ?\B  ?泯??????????"?? Q # 痂?  ? ' @\C# ?} h P 穰 A\ 3 ?泯B C<DE连F??????? ??++??vP.1)?6?Glkp?g?d^^??6 *I'PQ^gs??????<"+H<Q6[2c*j"lt??  @              ?"` ? '鹬 B\ 3 ?泯BCPDEF?????? ??? /P@ ?"` ? 鹭 C\  ??$攫???? ??????"??w ??  ? D\ # ?M?,琉??????????? ?  ?$D 0 ??Peptidyl transferaseF$??$ 鹭 E\  ???起???? ??????"??}, ? ??  痱 F\  ??焐???? ??????"??m? ??Chloramphenicol(50S,A)&?`  G\  ??H瑞????? ??????"??  ???,0Mechanism of action0 &?$f3鹦B H\?  ?d跟???D??????"??v ?$D 0??  ?t I\A# < ?P ?B J\B  ??D?????????  ? ?B K\B  ??D?????????  t? \ ? ????????藿h? ? ???TTr??ff?乔?????????___PPT10?i??滥?+D?' ????= @B +?0 ?瘅瘙`??  `鹞 `  ?? 责????? ??????"?? ? ????8___PPT10??N___PPT9?0( ???&0pharmacokinetics0 B&?$f3&?$f3&?$f3? ` ??疔?? ???????&f? ??x?0___PPT10??8___PPT9? ??Chloramphenicol may be administered either intravenously or orally It penetrate blood-brain barrier, placental barrier, blood-ocular barrier It is inactivated by conjugation with glucuronic acid in liver, secreted by the renal tubule.?&?ff"$ - @`??? ` ? ????????藿h? ? ???33?洙??33???y___PPT10?Y+D?' ????= @B +6?0 ]?帼d痦?  d痱 d ??(铕??? ??????"??< $  ??? 0Clinical uses0 &?$f3鸹 d ????? ??????"????l??x?0___PPT10??8___PPT9? 稹? Bacterial meningitis: meningococcal meningitis Rickettsial infections: typhus or Rocky Mountain spotted fever Eye infection: outer eye infection, intraocular infection, eyeball infection Anaerobic infection: peritoneal abscess, pelvic inflammation and peritonitis @?.&?ff"&?ff0  @`??? d ? ????????藿h? ? ???33?洙??33???y___PPT10?Y+D?' ????= @B +?0 瘌玄h??  h鹦 h ????? ??????"??? ?????8___PPT10??N___PPT9?0( ???"0Adverse effect0 T&?$?&?$?&?$?&?$f3? h ??T??? ??????"??? I1 ????8___PPT10??H___PPT9?*" ???Bone marrow depression Aplastic anemia Gray baby syndrome: poor feeding, depressed breathing, cardiovascular collapse, cyanosis and death \=?\?;&?ff""?V&?ffz @`??? h ? ????????藿h? ? ???TTr??ff?乔?????????___PPT10?i??例;?+D?' ????= @B +E?0 \?Pml痨?  l痄 l  ??????? ??????"??& ?????8___PPT10??N___PPT9?0( ???&0Drug resistance 0 X'?$f3&?$f3&?$f3'?$f3鹑 l ?????? ??????"???m ??x?0___PPT10??8___PPT9? 皎??Produce inactivator? acetyl coenzyme A transferase Membrane permeability is decreased, chloramphenicol penetrate the organism less"???&?ffH  % @`??? l ? ????????藿h? ? ???TTr??ff?乔?????????___PPT10?i?????+D?' ????= @B +?0 `? ??   鸩  ??0+??? ??????"??B??v?0___PPT10??6___PPT9? ??@Artificial Synthetic antibacterial drugs AA&?$` 7穰   ??????? ??????? 0! ??v?0___PPT10??6___PPT9? ??Section I Quinolones : &?$`  &?$` ?  ? ????????藿h? ? f????觋f?f???????y___PPT10?Y+D?' ????= @B +?0  衅穑?  ?  ????? ??????"??9%??v?0___PPT10??6___PPT9? ??The first generation : nalidixic acid, pipemidic acid The second generation: norfloxacin, ofloxacin, ciprofloxacin The third generation: sparfloxacin, levofloxacin, grepafloxacin The fourth generation: clinafloxacin, gatifloxacin. ?x&? `&?f3&? `?&?f3&? `?&?f3&? `&?f3    &     ?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10????Q|??0 瘐??  ?   ??????? ??????"??Y ?  鸨?SFluorequionlones: The second generation The third generation The fourth generation T?T&? `C?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???p?w9?0 P?? 疣?   ?  ??????? ???"??0??v?0___PPT10??6___PPT9? ???.0antibacterial action0 "0?&?$?  ??$a?? ???"??M%??x?0___PPT10??8___PPT9? ?^All of the quinolones are bactericidal First generation only has active against some gram-negative bacteria Second generation expend gram-negative bacteria spectrum Third generation have active against gram-positive organisms, chlamydia, mycoplasma, Legionella and Bacillus tuberculosis The fourth generation have active against anaerobic bacterium &_1?x_&?ffP    [ @`???  ? ????????藿h? ? f????觋f?f????????___PPT10?i??晒+D?' ????= @B +|?0 ?? ??   ?  ??Hs?? ??????}TZ ??v?0___PPT10??6___PPT9? ??? interfering with the action of DNA gyrase: gram-negative bacteria interfering with the action of topoisomerase IV: gram-positive bacteria ?,vv2vv?&?f3 '?$ff6#? !鹦   ??????? ?????? V ???  ?   ??|????? ??????"??8]??v?0___PPT10??6___PPT9? ??)Inhibit the replication of bacterial DNA **&?ff    ??T?????? ??????"??< ???,0Mechanism of action0 &?$??  ? ????????藿h? ? ???33?洙??33???y___PPT10?Y+D?' ????= @B +n?0 ???? ??   鹦   ??T????? ???????  ???  痱  ??% ?? precursor  &?f  p ??\H?????P   皙??:Purine0 pyrimidine nucleotide&?f.  皎  p ? ??"?0e???0e??????    B8CPDEF?????? ???????????????????????@ ?  狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??@A?BCD|E???????8tX?X(P@  ?#" ?? 鸠 p ??N?????? L ?? Glutamate  &?f皎 p # ??A??? ??? ?????? 0 ? 皎 p # ??A??? ??? ??????9P  痣? b  p ??? @?$D 0鸠 p ? ??????b  ?? Sulfonamides &?1'?皙 p  ??A ??? ?????? 0 r 鹭 p  ??U????? ??????"??{??????8___PPT10??N___PPT9?0( ???,0Mechanism of action0 F'?$f3&?$f3'?$f3皎 p # ??A??? ??? ?????? ]  ?  皎 p # ??A??? ??? ??????0 ? 皎 p # ??A??? ??? ??????0 ? ? p ? ????????藿h? ? ???TTr??ff?乔???????___PPT10????@?+??D?' ????= @B D?' ?????= @BA?%?( < +O%?( < +D?' =%(????D' =%(D窬' =?@B?B?BB%(D聒' =1?:Bvisible*?3>?B?style.visibility<?p????????%(D' =+襻4 8??CB0-#ppt_w/2BCB#ppt_xB*?3>B ppt_x<?p????????D' =+褓4 8??CB#ppt_yBCB#ppt_yB*?3>B ppt_y<?p????????+`?0 鹑帻t??  t痍 t  ??Y????? ??????"??jd 甬??<___PPT10??Z___PPT9?<4 ???"0Clinical uses 0 R'?$f3 &?$f3 ? '? $f3疝 t ??????? ???"?? Zj  ??&0??g ff ? t  ??Lv???? ??????"??I"??x?0___PPT10??8___PPT9? ??Systemic infections: oral and absorbable sulfonamides 2. Intestinal infection: oral and nonabsorbable sulfonamides 3. Wound infection: topical sulfonamides,???&?ffb < @`??? t ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10????跸?0 5??x鹋?  x痤 x  ??q????? ??????"??+ 8甬??<___PPT10??Z___PPT9?<4 ???"0adverse effect 0V'?$?&?$?$?? '? $?? x ??d??? ??????"??<&?W??v?0___PPT10??6___PPT9? ?O1. Crystalluria: crystallura, hematuria, obstruction adequate hydration and alkalinization of urine 2. Kernicterus: sulfonamides displace bilirubin from binding sites on serum albumin 3. Hypersensitivity: rashes, angioedema 4. Hemopoietic disturbances: Hemolytic anemia, Granulocytopenia thrombocytopenia LPx&?f3?&?ff &?ff   *  H  & @`??? x ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???? U?0 e?)|瘐?  |鸾 | ????? ??????"???I/ ??v?0___PPT10??6___PPT9? 馥?YContraindications: newborns and infants less than 2 months old as well as pregnant women0Z?&?f3?&?ff? | ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10?????芗?0 X??痂?  痤   ??T?????? ??????"??l H甬??<___PPT10??Z___PPT9?<4 ???&0drug resistance 0 R'?$f3&?$f3 ? '? $f3鸷  ????? ??????"??0????8___PPT10??H___PPT9?*" ??Increased PABA synthesis: overcome the inhibition of the dihydropteroate synthetase by the sulfas 2. Altered enzyme: decreased affinity for the sulfonamides 3. Decreased uptake: decreased permeability of membrane>??&?ff?&?ff,> ? @`???  ? ????????藿h? ? ???33?洙??33n?0 鹬????  ?   ??暗???? ??????"??W?X??v?0___PPT10??6___PPT9? ??Oral, absorbable agents &?$`鸶   ??瑚???? ??????"?? ??v?0___PPT10??6___PPT9? ??.Sulfisoxazole Sulfamethoxazole Sulfadiazine /?/&? `$ ?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10?????0 T?嘤?痄?  ?瓞 ? ??厉?? ??????"??& ????4___PPT10? ?B___PPT9?$ ?? Sulfisoxazole and sulfamethoxazole are used almost exclusively to treat urinary tract infections. Sulfadiazine achieves high concentrations in cerebrospinal fluid, therefore it has preventative and therapeutic effective against Epidemic meningitis(? &?ff. ? ? ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10??? ∞?0 9???鹕?  ?   ??P流???? ??????"??GX??v?0___PPT10??6___PPT9? ??Oral nonabsorbable agents &?$`  痫  ??t索?? ??????"??d? ??v?0___PPT10??6___PPT9? 鹱?i Sulfasalazine is widely used in ulcerative colitis, enteritis, and other inflammatory bowel disease. 0j?&?f3?&?ff Y?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???i骱X?0 鹄p???  ?   ??茉???? ??????"?? X??v?0___PPT10??6___PPT9? ??Topical Agents&?$`瓞  ??嘭?? ??????"??" ??v?0___PPT10??6___PPT9? ??(Sodium sulfacetamide Mafenide acetate ))&? `,  ?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10?????0?0 E?`?鹫?  ?  ??拜?? ??????"???| ??v?0___PPT10??6___PPT9? ?? Sodium sulfacetamide ophthalmic solution or ointment is effective treatment for bacterial conjunctivitis and as adjunctive therapy for trachoma. Mafenide acetate is used topically to prevent bacterial colonization and infection of burn wounds. 0?&?f3?&?ff4 ?\?  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???屑????0 痦P? ??   ?    ?? 眵???? ??????"??Z ??v?0___PPT10??6___PPT9? ?? Trimethoprim &?$` 鹄   ??铟?? ??????"??z?????8___PPT10??L___PPT9?.& ??V1. The antibacterial spectrum is similar to that of sulfamethoxazole It inhibited dihydrofolate reductase It is used alone in acute urinary tract infections and in the treatment of bacterial prostatitis It induce megaloblastic anemia, leukopenia, and granulocytopenia It altered dihydrofolate reductase, resulting in drug resistancePNx x&?f3?&?ff &?ff<  W      @`???   ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???Pm?0 ,?@?鸺?  ?  ??<喵?? ??????"??ZJ.??v?0___PPT10??6___PPT9? ??Co-trimoxazole&?$? 瘊  ??|?? ??????"??M\?] ????8___PPT10??N___PPT9?0( 鹇?Co-trimoxazole is combination of trimethoprim- sulfamethoxazole It shows greater antimicrobial activity than equivalent quantities of either drug used alone It inhibits two sequential steps in the synthesis of tetrahydrofolic acidL/???F&?ff?&?ffP  ? @`???  ? ????????藿h? ? ???TTr??ff?乔??????8?0___PPT10???0 ?N?0 皎须???  ?皙 ? ????????9Y ??" 鹭 ? ???(??????i?l ??PABA + Pteridine&? f 鹩 ? ??H-?????/? ??Dihydropteroic acid&? f痖 ? ????????O U ??Dihydropteroate synthase$??$鹜  ? ??x6?????m ?  ?? Dihydrofolate&? f   ? ?????? ??"?? 4  ??Dihydrofolate reductase(DHFR)$??$ 鹦  ? ??p??????S ?  ??Tetrahydrofolate&? f穑  ? ? ??????0?>? ?? precursor  &? f  ? ??\H?????A ? 皙??:Purine0 pyrimidine nucleotide&? f.  皎 ? ? ??"?0e???0e??????    B8CPDEF?????? ???????????????????????@ ?  狭?怂 8c8c     ??????1??瘗??? d0u0盱?@T?????y?2 NP'p????'p??@A?BCD|E???????8tX?X(P@  ?#" ??  W鸠 ? ????????O ? ?? Glutamate  &?f皎 ? # ??A??? #??? ??????? 0   #皎 ? # ??A??? $??? ??????D  $皎 ? # ??A??? %??? ??????e7 ? U %皎 ? # ??A??? &??? ??????r? ?  &皎 ? # ??A??? '??? ???????P [ '?? b  ? ? ?$D 0? ? ? ??????b ??v?0___PPT10??6___PPT9? ??sulfamethoxazole &?1'?皙 ?  ??A (??? ?????? 0 r (鸾? ? P l  ? ? ?P ? ?$D 0瘐 ? ? ??PZ???? ` l  ??Trimethoprim (TMP)D &?1'?&? 1'?&?1'? ? ?  A o P  ? ? ? ????????藿h? ? ???TTr??ff?乔??????F ?> ___PPT10? ?y?`9?+^YID耱 ' ????= @B D癍 ' ?????= @BA?%?( < +O%?( < +D?' =%(????D' =%(D窬' =?@B?B?BB%(D聒' =1?:Bvisible*?3>?B?style.visibility<??????????%(D' =+襻4 8??CB0-#ppt_w/2BCB#ppt_xB*?3>B ppt_x<??????????D' =+褓4 8??CB#ppt_yBCB#ppt_yB*?3>B ppt_y<??????????D?' =%(????D' =%(D窬' =?@B?B?BB%(D聒' =1?:Bvisible*?3>?B?style.visibility<??????????%(D' =+襻4 8??CB0-#ppt_w/2BCB#ppt_xB*?3>B ppt_x<??????????D' =+褓4 8??CB#ppt_yBCB#ppt_yB*?3>B ppt_y<??????????+?0 0?瓞?  ?  ?? b?? ??????"??,K ??v?0___PPT10??6___PPT9? ????4. Co-trimoxazole is used to treat upper respiratory infection, urinary tract infection ? intestinal infection ?typhoid fever 5. 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